Chemical Stability of Insulin. 1. Hydrolytic Degradation During Storage of Pharmaceutical Preparations Jens BrangeLiselotte Langkj\sgmaelig;rAage Vølund OriginalPaper Pages: 715 - 726
Chemical Stability of Insulin. 2. Formation of Higher Molecular Weight Transformation Products During Storage of Pharmaceutical Preparations Jens BrangeSvend HavelundPhilip Hougaard OriginalPaper Pages: 727 - 734
Derivatives of 4-(2-N,N-Di-n-propylaminoethyl)-5-hydroxyindole: Synthesis and Pharmacological Effects Joseph G. CannonIoannis RoufosJohn Paul Long OriginalPaper Pages: 735 - 738
Structural Modification Study of Anthracyclinones: Synthesis and Biological Activity of Several Derivatives of η-Pyrromycinone Dun-Fu LiuHui XiongChia-Chung Cheng OriginalPaper Pages: 739 - 742
Improved Delivery Through Biological Membranes. XLV. Synthesis, Physical-Chemical Evaluation, and Brain Uptake Studies of 2-Chloroethyl Nitrosourea Delivery Systems Krishnaswamy RaghavanThorsteinn LoftssonNicholas Bodor OriginalPaper Pages: 743 - 749
Parenteral Formulation of the Kappa Agonist Analgesic, DuP 747, via Micellar Solubilization Munir A. HussainLei-Shu WuArthur R. Hurwitz OriginalPaper Pages: 750 - 752
Acceleration of Heat Transfer in Vial Freeze-Drying of Pharmaceuticals. II. A Fluid Cushion Device Samuel H. YalkowskySuresh D. Patel OriginalPaper Pages: 753 - 758
Microencapsulation of Solid Dispersions: Release of Griseofulvin from Griseofulvin:Phospholipid Coprecipitates in Microspheres Gopi K. VudathalaJames A. Rogers OriginalPaper Pages: 759 - 763
The Pharmacokinetics of Pulmonary-Delivered Insulin: A Comparison of Intratracheal and Aerosol Administration to the Rabbit Paul ColthorpeStephen J. FarrDavid Wyatt OriginalPaper Pages: 764 - 768
Conjunctival Penetration of Insulin and Peptide Drugs in the Albino Rabbit Eiji HayakawaDu-Shieng ChienVincent H. L. Lee OriginalPaper Pages: 769 - 775
Immobilization of Active Urokinase on Albumin Microspheres: Use of a Chemical Dehydrant and Process Monitoring Kumaril BhargavaHoward Y. Ando OriginalPaper Pages: 776 - 781
Macrophage Activation by Polymeric Nanoparticles of Polyalkylcyanoacrylates: Activity Against Intracellular Leishmania donovani Associated with Hydrogen Peroxide Production Rogério GasparVeronique PréatMichel Roland OriginalPaper Pages: 782 - 787
The Mobile Order Theory Versus UNIFAC and Regular Solution Theory-Derived Models for Predicting the Solubility of Solid Substances Paul RuelleMichel BuchmannUlrich W. Kesselring OriginalPaper Pages: 788 - 791
Cholesterol (Thermodynamic) Activity Determinations in Bile Salt–Lecithin–Cholesterol Systems and Cholesterol-Rich Liquid Crystalline Mesophase Formation Uday K. JainWilliam I. HiguchiNorman A. Mazer OriginalPaper Pages: 792 - 799
Plasma Concentration Clamping in the Rat Using a Computer-Controlled Infusion Pump Lars L. GustafssonWilliam F. EblingSteven L. Shafer OriginalPaper Pages: 800 - 807
Stability of the New Anticancer Platinum Analogue 1,2-Diaminomethyl-Cyclobutane-Platinum(II)-Lactate (Lobaplatin; D19466) in Intravenous Solutions Henk-Jan GuchelaarDonald R. A. UgesNanno H. Mulder OriginalPaper Pages: 808 - 811
Simultaneous Microdetermination of Rifampin, Deacetylrifampin, Isoniazid, and Acetylisoniazid in Plasma by Liquid Chromatography with Dual Electrochemical and Spectrophotometric Detection Adnan El-YazigiDale A. Raines OriginalPaper Pages: 812 - 816
Comparison of Azone and Hexamethylene Lauramide in Toxicologic Effects and Penetration Enhancement of Cimetidine in Rabbit Eyes I. Maged IsmailChi-Chu ChenDiane D.-S. Tang-Liu Note Pages: 817 - 821
Pharmacokinetics of Oral 2′,3′-Dideoxyinosine in Rats M. Guillaume WientjesJessie L.-S. Au Note Pages: 822 - 825
Opportunities for Integration of Pharmacokinetics, Pharmacodynamics, and Toxicokinetics in Rational Drug Development Carl C. PeckWilliam H. BarrAvraham Yacobi Conference Report Pages: 826 - 833