Functional Expression and Localization of P-glycoprotein in the Central Nervous System: Relevance to the Pathogenesis and Treatment of Neurological Disorders Gloria LeeReina Bendayan ReviewPaper Pages: 1313 - 1330
The Role of Metabolites in Bioequivalence Kamal K. MidhaMaureen J. RawsonJohn W. Hubbard Commentary Pages: 1331 - 1344
A Compartment Model for the Membrane-Coated Fiber Technique Used for Determining the Absorption Parameters of Chemicals into Lipophilic Membranes Xin-Rui XiaRonald E. BaynesJim E. Riviere OriginalPaper Pages: 1345 - 1352
Use of Biophysical Characterization in Preformulation Development of a Heavy-Chain Fragment of Botulinum Serotype B: Evaluation of Suitable Purification Process Conditions Frank K. Bedu-AddoCatharine JohnsonSiddharth J. Advant OriginalPaper Pages: 1353 - 1361
Effects of the Chemical Structure and the Surface Properties of Polymeric Biomaterials on Their Biocompatibility You-Xiong WangJohn L. RobertsonRichard O. Claus OriginalPaper Pages: 1362 - 1373
Characterization and In Vivo Study of Sustained-Release Formulation of Human Growth Hormone Using Sodium Hyaluronate Sei Kwang HahnSun Jin KimDuk Hee Kim OriginalPaper Pages: 1374 - 1381
In Situ Transport of Vinblastine and Selected P-glycoprotein Substrates: Implications for Drug-Drug Interactions at the Mouse Blood-Brain Barrier Salvatore CisterninoChristophe RousselleJean-Michel Scherrmann OriginalPaper Pages: 1382 - 1389
Porcine Ear Skin as a Model for the Assessment of Transdermal Drug Delivery to Premature Neonates Nabila SekkatYogeshvar N. KaliaRichard H. Guy OriginalPaper Pages: 1390 - 1397
Transport Characteristics of Fexofenadine in the Caco-2 Cell Model Niclas PetriChrister TannergrenHans Lennernäs OriginalPaper Pages: 1398 - 1404
Susceptibility to Lipase-Mediated Digestion Reduces the Oral Bioavailability of Danazol After Administration as a Medium-Chain Lipid-Based Microemulsion Formulation Christopher J. H. PorterAnn Marie KaukonenWilliam N. Charman OriginalPaper Pages: 1405 - 1412
Influence of the Type of Surfactant and the Degree of Dispersion on the Lymphatic Transport of Halofantrine in Conscious Rats Ditte M. KarpfRené HolmAnette Müllertz OriginalPaper Pages: 1413 - 1418
Solvent Exchange Method: A Novel Microencapsulation Technique Using Dual Microdispensers Yoon YeoAlvin U. ChenKinam Park OriginalPaper Pages: 1419 - 1427
Physicochemical Parameters Associated with Nanoparticle Formation in the Salting-Out, Emulsification-Diffusion, and Nanoprecipitation Methods Sergio Galindo-RodriguezEric AllémannEric Doelker OriginalPaper Pages: 1428 - 1439
Inverse Gas Chromatography: Investigating Whether the Technique Preferentially Probes High Energy Sites for Mixtures of Crystalline and Amorphous Lactose Helen E. NewellGraham Buckton OriginalPaper Pages: 1440 - 1444
Hydrophilic Microspheres from Water-in-Oil Emulsions by the Water Diffusion Technique Michele TrottaDaniela ChirioElena Peira OriginalPaper Pages: 1445 - 1449
Identification of Stabilized Dynorphin Derivatives for Suppressing Tolerance in Morphine-Dependent Rats Suliman I. Al-FayoumiBoglarka BrugosGünther Hochhaus OriginalPaper Pages: 1450 - 1456
Evaluating Barriers to Bioavailability in Vivo: Validation of a Technique for Separately Assessing Gastrointestinal Absorption and Hepatic Extraction Laura LetendreMark ScottBruce Aungst OriginalPaper Pages: 1457 - 1462
Population Dose-Response Model for Tadalafil in the Treatment of Male Erectile Dysfunction Alexander StaabChristiane TillmannIñaki F. Trocóniz OriginalPaper Pages: 1463 - 1470
Enhancement of Transfection Efficiency Through Rapid and Noncovalent Post-PEGylation of Poly(Dimethylaminoethyl Methacrylate)/DNA Complexes Sabine PirottonCaroline MullerMartine Raes OriginalPaper Pages: 1471 - 1479
How Well Can an Idiotope Peptide Mimic Replace Its Parent Idiotype in a Synthetic Peptide Vaccine? James S. CavenaughHsu-Kun WangJames N. Herron OriginalPaper Pages: 1480 - 1488
Evidence for Modulation of P-glycoprotein-Mediated Efflux by Methoxypolyethylene Glycol-block-Polycaprolactone Amphiphilic Diblock Copolymers Jason ZastreJohn JacksonHelen Burt OriginalPaper Pages: 1489 - 1497
The Mechanism of Protraction of Insulin Detemir, a Long-Acting, Acylated Analog of Human Insulin Svend HavelundAnne PlumPeter Kurtzhals OriginalPaper Pages: 1498 - 1504
Insertion and Partition of Sodium Taurocholate into Egg Phosphatidylcholine Vesicles Karine AndrieuxLaura ForteCécile Grabielle-Madelmont OriginalPaper Pages: 1505 - 1516