Insulin Fragments as a Carrier for Peptide Delivery Across the Blood–Brain Barrier Makoto FukutaHiroaki OkadaHajime Toguchi OriginalPaper Pages: 1681 - 1688
Transsynovial Drug Distribution: Synovial Mean Transit Time of Diclofenac and Other Nonsteroidal Antiinflammatory Drugs William F. ElmquistKeith K. H. ChanRonald J. Sawchuk OriginalPaper Pages: 1689 - 1697
The Effect of Cyclodextrins on the Stability of Peptides in Nasal Enzymic Systems William J. IrwinAnil K. DwivediMichael J. Dey OriginalPaper Pages: 1698 - 1703
Mechanism of Optical Isomerization of(S)-N-[1-(2-Fluorophenyl)-3,4,6,7-tetrahydro-4-oxopyrrolo[3,2,1-jk] [l,4]-benzodiazepine-3-y1]-1H-indole-2-carboxamide (FK480) in Soft Capsules Containing Polyethylene Glycol 400 and Glycerol Shinichi FukuyamaNoriaki KiharaTsutomu Yasuda OriginalPaper Pages: 1704 - 1706
Menthol-β-D-Glucuronide: A Potential Prodrug for Treatment of the Irritable Bowel Syndrome Harold W. Nolen IIIDavid R. Friend OriginalPaper Pages: 1707 - 1711
Aqueous Stability of Human Epidermal Growth Factor 1-48 Richard I. SenderoffScott C. WoottonGalen W. Radebaugh OriginalPaper Pages: 1712 - 1720
Is Stability Prediction Possible for Protein Drugs? Denaturation Kinetics of β- Galactosidase in Solution Sumie YoshiokaYukio AsoS. Kojima OriginalPaper Pages: 1721 - 1725
Natriuretic Peptide-Potentiating Actions of Neutral Endopeptidase Inhibition in Rats with Experimental Heart Failure Masato YasuharaMasayuki YamaguchiRyohei Hori OriginalPaper Pages: 1726 - 1730
Targeted Gene Delivery to Alveolar Macrophages via Fc Receptor-Mediated Endocytosis Yongyut RojanasakulLi Ying WangJiahorng Liaw OriginalPaper Pages: 1731 - 1736
The Relation Between Swelling Properties and Enzymatic Degradation of Azo Polymers Designed for Colon-Specific Drug Delivery Guy Van den MooterCelest SamynRenaat Kinget OriginalPaper Pages: 1737 - 1741
Effect of Current Magnitude and Drug Concentration on lontophoretic Delivery of Octreotide Acetate (Sandostatin®) in the Rabbit David T.-W. LauJohn W. SharkeyFrancis L. S. Tse OriginalPaper Pages: 1742 - 1746
Improving the Sensitivity of in Vitro Skin Penetration Experiments Gerald B. KastingThomas G. FilloonMichael P. Meredith OriginalPaper Pages: 1747 - 1754
The Effects of Bile Salts and Lipids on the Physicochemical Behavior of Gemfibrozil Paul E. LunerSuresh R. BabuGalen W. Radebaugh OriginalPaper Pages: 1755 - 1760
Characteristics of Ceftibuten Uptake into Caco-2 Cells Noriyuki MuranushiKazutoshi HorieKoichiro Hirano OriginalPaper Pages: 1761 - 1765
Effect of 2-Hydroxypropyl-β-cyclodextrin on Crystallization and Polymorphic Transition of Nifedipine in Solid State Fumitoshi HirayamaZheng WangKaneto Uekama OriginalPaper Pages: 1766 - 1770
Comparison of the Transport Characteristics of D- and L-Methionine in a Human Intestinal Epithelial Model (Caco-2) and in a Perfused Rat Intestinal Model Lixing ZhengJiyue ChenMing Hu OriginalPaper Pages: 1771 - 1776
Transport of β-Estradiol in Freshly Excised Human Skin in Vitro: Diffusion and Metabolism in Each Skin Layer Puchun LiuWilliam I. HiguchiWilliam R. Good OriginalPaper Pages: 1777 - 1784
The Role of Rheological Properties in Mucociliary Transport by Frog Palate Ciliated Model Danny M. YuGordon L. AmidonArthur H. Goldberg OriginalPaper Pages: 1785 - 1791
Formation and Characterization of Cisplatin-Loaded Poly(benzyl 1-glutamate) Microspheres for Chemoembolization Chun LiDavid J. YangSidney Wallace OriginalPaper Pages: 1792 - 1799
Surface Modification of Poly(lactide-co-glycolide) Nanospheres by Biodegradable Poly(lactide)-Poly(ethylene glycol) Copolymers Snjezana StolnikSusan E. DunnLisbeth Illum OriginalPaper Pages: 1800 - 1808
Effect of Electroporation on Transdermal lontophoretic Delivery of Luteinizing Hormone Releasing Hormone (LHRH) in Vitro D. Bommi BommannanJanet TamadaRussell O. Potts OriginalPaper Pages: 1809 - 1814
Enantioselective Kinetics of Verapamil and Norverapamil in Isolated Perfused Rat Livers Reza MehvarJames M. ReynoldsJames A. Longstreth OriginalPaper Pages: 1815 - 1819
Effect of Perfusate pH on Reduction of Quinidine Capillary Permeability by Albumin in Isolated Perfused Rat Heart Denis J. MorganCao Ling Xu OriginalPaper Pages: 1820 - 1824
The Use of Multiple Doses and Pharmacodynamic System Analysis to Distinguish Between Dispositional Delays and Time-Variant Pharmacodynamics Marc R. GastonguaySorell L. Schwartz OriginalPaper Pages: 1825 - 1828
Effect of Substituted Benzoylglycines (Hippurates) and Phenylacetylglycines on p-Aminohippurate Transport in Dog Renal Membrane Vesicles Frans G. M. RusselWim G. Vermeulen OriginalPaper Pages: 1829 - 1833
Rapid Temporal Control of Transdermal Drug Delivery by Electroporation Mark R. PrausnitzUwe PliquettJames C. Weaver Note Pages: 1834 - 1837